Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50067581'
LigandPNGBDBM50067581((S)-2-{[2'-Methyl-5-(pyridin-3-ylaminomethyl)-biph...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067581((S)-2-{[2'-Methyl-5-(pyridin-3-ylaminomethyl)-biph...)
Affinity DataIC50:  0.420nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed