Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50076794'
LigandPNGBDBM50076794(CHEMBL276602 | Lithium; (S)-2-({5-[5-(4-isopropyl-...)
Affinity DataIC50:  2.90nMAssay Description:In vitro inhibitory activity of the compound was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50076794(CHEMBL276602 | Lithium; (S)-2-({5-[5-(4-isopropyl-...)
Affinity DataEC50:  0.780nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed