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Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50082915'
LigandPNGBDBM50082915((S)-2-({5-[((S)-1-Cyclohexylmethyl-2-o-tolylsulfan...)
Affinity DataIC50:  0.420nMAssay Description:In vitro inhibitory activity against Farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed