Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50106863'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Lgci
Curated by ChEMBL
Lgci
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of farnesyltransferase activity against H-RasMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Lgci
Curated by ChEMBL
Lgci
Curated by ChEMBL
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of farnesyltransferase activity against K-RasMore data for this Ligand-Target Pair