Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50106869'
LigandPNGBDBM50106869(CHEMBL102435 | [1-(3-Benzyl-3H-imidazol-4-ylmethyl...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of farnesyltransferase activity against H-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106869(CHEMBL102435 | [1-(3-Benzyl-3H-imidazol-4-ylmethyl...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of farnesyltransferase activity against K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed