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Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50108070'
LigandPNGBDBM50108070(2-[4-(2-Amino-3-mercapto-propylamino)-benzoylamino...)
Affinity DataKi:  785nMAssay Description:Inhibition of recombinant FTase (unknown origin)-mediated K-Ras4B model peptide KKKKKKSK(Dans)TKCVIM farnesylation by fluorescence plate reader analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed