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Found 3 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50407296'
LigandPNGBDBM50407296(CHEMBL2052018 | L-731735)
Affinity DataIC50:  18nMAssay Description:Activity against bovine FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50407296(CHEMBL2052018 | L-731735)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407296(CHEMBL2052018 | L-731735)
Affinity DataIC50:  20nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed