Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50493656'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi
Curated by ChEMBL
'Al. I. Cuza' University Of Iasi
Curated by ChEMBL
Affinity DataIC50: 4.35E+4nMAssay Description:Inhibition of recombinant human farnesyltransferase using Dansyl-GCVLS as substrate measured for 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair