TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]-PDBU ligand from recombinant protein kinase C (baculovirus)More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]PDBu from mouse recombinant PKCalpha expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMpH: 7.4Assay Description:Inhibition of [3H]PDBu binding to recombinant protein kinase C alpha was determined at pH 7.4, 37 degree C for 5 minMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity for Protein kinase C alpha C1a or C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 402nM ΔG°: -35.6kJ/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair