Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Protein kinase C beta type' and Ligand = 'BDBM50185931'
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed