Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PKCtheta using Histone H1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human PKCtheta using Histone H1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PKCtheta (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PKCtheta (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Binding constant for PRKCQ kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Binding constant for PRKCQ kinase domainMore data for this Ligand-Target Pair