Found 2 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP4' and Ligand = 'BDBM50250875'
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
University Of Oslo
Curated by ChEMBL
University Of Oslo
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
University Of Oslo
Curated by ChEMBL
University Of Oslo
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PARP4 using NAD+ as substrate by fluorescence assayMore data for this Ligand-Target Pair