Found 4 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP4' and Ligand = 'BDBM50316226'
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Irbm/Merck Research Laboratories
Curated by ChEMBL
Irbm/Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of human v-PARP catalytic domain by trichloroacetic acid precipitation assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Irbm/Merck Research Laboratories
Curated by ChEMBL
Irbm/Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 446nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Irbm/Merck Research Laboratories
Curated by ChEMBL
Irbm/Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 447nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Irbm/Merck Research Laboratories
Curated by ChEMBL
Irbm/Merck Research Laboratories
Curated by ChEMBL
Affinity DataKd: 272nMAssay Description:Binding affinity to PARP4 (unknown origin) assessed as apparent dissociation constantMore data for this Ligand-Target Pair