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Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM50277163'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Alma Mater Studiorum-University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50277163(CHEMBL4177374)
Affinity DataIC50:  4.84E+5nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed