Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM50400625'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa

Curated by ChEMBL
LigandPNGBDBM50400625(CHEMBL2203469)
Affinity DataKi:  1.74E+4nMAssay Description:Irreversible inhibition of human TG2 using AL5 as substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa

Curated by ChEMBL
LigandPNGBDBM50400625(CHEMBL2203469)
Affinity DataIC50:  62nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed