Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50274114' TargetProteinase-activated receptor 2(Homo sapiens (Human))
Shanghai Jiao Tong University
Curated by ChEMBL
Shanghai Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: <2.5nMAssay Description:Antagonist activity at human PAR2More data for this Ligand-Target Pair
3D Structure (crystal)TargetProteinase-activated receptor 2(Homo sapiens (Human))
Shanghai Jiao Tong University
Curated by ChEMBL
Shanghai Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Antagonist activity at PAR2 in human 1321N1 cells assessed as inhibition of trypsin-induced intracellular calcium flux pretreated for 60 mins followe...More data for this Ligand-Target Pair
