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Found 3 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM50034417'
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50034417(4-Amino-N-[1,3,4]thiadiazol-2-yl-benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The University Of Texas

Curated by ChEMBL
LigandPNGBDBM50034417(4-Amino-N-[1,3,4]thiadiazol-2-yl-benzenesulfonamid...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Akt phosphorylation in human BxPC3 cells by Western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The University Of Texas

Curated by ChEMBL
LigandPNGBDBM50034417(4-Amino-N-[1,3,4]thiadiazol-2-yl-benzenesulfonamid...)
Affinity DataKd:  450nMAssay Description:Inhibition of pleckstrin homology domain of AKT by surface plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed