Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM50304371'
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50304371(CHEMBL611216 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The University Of Texas

Curated by ChEMBL
LigandPNGBDBM50304371(CHEMBL611216 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt phosphorylation in human BxPC3 cells by Western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed