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Found 3 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase [1-123]' and Ligand = 'BDBM50304370'
TargetRAC-alpha serine/threonine-protein kinase [1-123](Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM50304370(CHEMBL593946 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKi: >5.00E+4nMAssay Description:SPR interaction analyses were performed with a Biacore 2000, using Biacore 2000 Control Software v3.2 and BIAevaluation v4.1 analysis software (Biaco...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [1-123](Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM50304370(CHEMBL593946 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of AKT was measured by Western blots using specific antibodies against phospho-Ser473-AKT in HT-29 lung cancer cells. Inhibition of the ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [1-123](Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM50304370(CHEMBL593946 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKd:  1.02E+4nMAssay Description:SPR interaction analyses were performed with a Biacore 2000, using Biacore 2000 Control Software v3.2 and BIAevaluation v4.1 analysis software (Biaco...More data for this Ligand-Target Pair
In DepthDetails US Patent