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Found 1 Enz. Inhib. hit(s) with Target = 'RAC-beta serine/threonine-protein kinase' and Ligand = 'BDBM126605'
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM126605(US8772283, 49)
Affinity DataIC50:  0.420nMpH: 7.5Assay Description:Preparation of AKT1 and AKT2 and measurement of in vitro inhibitory activity of the above-mentioned compounds against AKT1 and AKT2 kinase activity w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent