Found 2 Enz. Inhib. hit(s) with Target = 'Receptor tyrosine-protein kinase erbB-2' and Ligand = 'BDBM50390489'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of ERBB2 autophosphorylation Thr 1139 residue in human BT474 cells at 2 to 14 uM after 12 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKd: 2.90E+3nMAssay Description:Binding affinity to full-lenght/His-tagged ERBB2 UV-vis emission spectroscopyMore data for this Ligand-Target Pair