Found 1 Enz. Inhib. hit(s) with Target = 'Receptor tyrosine-protein kinase erbB-3' and Ligand = 'BDBM50029668'
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Xi'An Jiaotong University
Curated by ChEMBL
Xi'An Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair