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Found 2 Enz. Inhib. hit(s) with Target = 'Receptor-interacting serine/threonine-protein kinase 1 [8-327]' and Ligand = 'BDBM530216'
TargetReceptor-interacting serine/threonine-protein kinase 1 [8-327](Homo sapiens (Human))
Denali Therapeutics

US Patent
LigandPNGBDBM530216(Preparation of 4-[(4R)-3,3-difluoro-4-methyl-1-pyr...)
Affinity DataIC50: <100nMAssay Description:Test compounds were serially diluted in DMSO at 100 fold final concentrations in the assay (1% DMSO final). In each well of a 384-well Plate were dis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1 [8-327](Homo sapiens (Human))
Denali Therapeutics

US Patent
LigandPNGBDBM530216(Preparation of 4-[(4R)-3,3-difluoro-4-methyl-1-pyr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Test compounds were serially diluted in DMSO at 100 fold final concentrations in the assay (1% DMSO final). In each well of a 384-well Plate were dis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent