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Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50064254'
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataIC50:  82nMAssay Description:Inhibition of binding to retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  13nMAssay Description:Transcriptional activation of retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  27nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed