Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50132584'
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132584((2Z,4E,6Z)-7-[3,5-Di-tert-butyl-2-(2,2-difluoro-et...)
Affinity DataKi:  11nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132584((2Z,4E,6Z)-7-[3,5-Di-tert-butyl-2-(2,2-difluoro-et...)
Affinity DataEC50:  3.40nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed