Found 7 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-beta' and Ligand = 'BDBM50032667'
Affinity DataKi: 191nMAssay Description:Binding affinity towards recombinantly expressed Retinoic acid receptor RXR-beta in baculoviral sysytem, by using 5 nM [3H]-targretin in a competitiv...More data for this Ligand-Target Pair
Affinity DataEC50: 213nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 191nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 213nMAssay Description:Effective concentration against retinoid receptor isoform (RXR beta) expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 213nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair
Affinity DataKd: 232nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair