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Found 2 Enz. Inhib. hit(s) with Target = 'Rhodopsin kinase GRK1' and Ligand = 'BDBM283997'
TargetRhodopsin kinase GRK1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM283997(E23 | US10023564, Example 23)
Affinity DataIC50:  6.70E+4nMpH: 7.0Assay Description:GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRhodopsin kinase GRK1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM283997(E23 | US10023564, Example 23)
Affinity DataIC50:  8.30E+4nMAssay Description:Inhibition of GRK1 (unknown origin) preincubated for 10 mins followed by peptide substrate and ATP addition measured after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed