Affinity DataIC50: 4.60nMAssay Description:Inhibition of human GRK7 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human GRK7 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Binding constant for GRK7 kinase domainMore data for this Ligand-Target Pair