Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'STE20/SPS1-related proline-alanine-rich protein kinase' and Ligand = 'BDBM2579'
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  14.4nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  17.2nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  130nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed