Found 3 Enz. Inhib. hit(s) with Target = 'STE20/SPS1-related proline-alanine-rich protein kinase' and Ligand = 'BDBM2579'
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 14.4nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 17.2nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair