Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Sarcoplasmic/endoplasmic reticulum calcium ATPase 1' and Ligand = 'BDBM50242014'
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rattus norvegicus)
Centre Of Experimental Medicine

Curated by ChEMBL
LigandPNGBDBM50242014(CHEMBL464006 | Morusin | Morusin, 3 | TCMDC-124149...)
Affinity DataIC50:  2.87E+4nMAssay Description:Inhibition of SERCA1 in rat INS-1E cells assessed as reduction in cell viability incubated for 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Centre Of Experimental Medicine

Curated by ChEMBL
LigandPNGBDBM50242014(CHEMBL464006 | Morusin | Morusin, 3 | TCMDC-124149...)
Affinity DataIC50:  4.36E+4nMAssay Description:Inhibition of SERCA1 in NewZealand rabbit skeletal muscle SR vesicles using ATP as substrate incubated for 2 mins followed by Ca2+ addition by NADH c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed