Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase/endoribonuclease IRE1' and Ligand = 'BDBM31085'
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
Ambit Biosciences

Curated by ChEMBL
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)
Affinity DataKd:  6.00E+3nMAssay Description:Binding constant for ERN1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed