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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase B-raf' and Ligand = 'BDBM50121690'
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50121690(CHEMBL3616960)
Affinity DataIC50:  668nMAssay Description:Inhibition of BRAF V599E mutant (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50121690(CHEMBL3616960)
Affinity DataIC50:  5.96E+3nMAssay Description:Inhibition of BRAF (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed