Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase B-raf' and Ligand = 'BDBM50514785'
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)
Affinity DataKd:  2nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)
Affinity DataKd:  2.40nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed