Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1' and Ligand = 'BDBM50149481'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50149481(5-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50:  237nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 1 (Chk1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed