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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk2' and Ligand = 'BDBM50256044'
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity in rat uterus by uterotonic assayMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Chk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed