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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase D1' and Ligand = 'BDBM50324322'
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324322(4-(2-cyclohexylaminopyridin-4-yl)-6-(piperazin-1-y...)
Affinity DataIC50:  1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324322(4-(2-cyclohexylaminopyridin-4-yl)-6-(piperazin-1-y...)
Affinity DataEC50:  115nMAssay Description:Inhibition of PKD1 assessed as inhibition of HDAC5 neuclear exportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed