Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase ICK' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 38.6nMAssay Description:Inhibition of human LCK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of ICK (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 53.3nMAssay Description:Inhibition of human LCK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair