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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK1' and Ligand = 'BDBM8053'
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM8053(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 24 | 4...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM8053(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 24 | 4...)
Affinity DataIC50:  5.00E+3nMpH: 7.5 T: 2°CAssay Description:D. melanogaster Polo kinase assays were performed as previously described40, using baculovirus-expressed Polo kinase. Enzyme was immunoprecipitated u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed