Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase RIO2' and Ligand = 'BDBM50550133'
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50550133(CHEMBL4754518)
Affinity DataIC50:  6.60E+3nMAssay Description:Displacement of fluorescent tracer K5 from N-terminal full-length NanoLuc-fused RIOK2 (unknown origin) expressed in HEK293 cells using NanoGlo substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50550133(CHEMBL4754518)
Affinity DataIC50:  6.60E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed