Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase STK11' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase STK11(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 48.7nMAssay Description:Inhibition of human LKB1 using LSNLYHQGKFLQTFCGSPLYRRR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase STK11(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 70.9nMAssay Description:Inhibition of human LKB1 using LSNLYHQGKFLQTFCGSPLYRRR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase STK11(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 61nMAssay Description:Binding constant for LKB1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase STK11(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 61nMAssay Description:Binding constant for full-length LKB1More data for this Ligand-Target Pair