Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-3' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 0.0890nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 0.0980nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 0.121nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 0.510nMAssay Description:Binding constant for PIM3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 0.510nMAssay Description:Binding constant for PIM3 kinase domainMore data for this Ligand-Target Pair