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Found 4 Enz. Inhib. hit(s) with Target = 'Serine protease 1' and Ligand = 'BDBM17279'
TargetSerine protease 1(Bos taurus (bovine))
Berlex

LigandPNGBDBM17279(2-(5-carbamimidoyl-2-hydroxyphenoxy)-6-[3-(4,5-dih...)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17279(2-(5-carbamimidoyl-2-hydroxyphenoxy)-6-[3-(4,5-dih...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibitory constant against bovine trypsin for general specificity against serine proteasesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex

LigandPNGBDBM17279(2-(5-carbamimidoyl-2-hydroxyphenoxy)-6-[3-(4,5-dih...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibitory potency was measured against bovine trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Berlex

LigandPNGBDBM17279(2-(5-carbamimidoyl-2-hydroxyphenoxy)-6-[3-(4,5-dih...)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair