Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Serine protease hepsin' and Ligand = 'BDBM525256'
TargetSerine protease hepsin(Human)
University of British Columbia

LigandChemical structure of BindingDB Monomer ID 525256BDBM525256(N-0438 | (H)Arg-Glu-Phe-Arg-kbt)
Affinity DataKi:  0.520nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
University of British Columbia

LigandChemical structure of BindingDB Monomer ID 525256BDBM525256(N-0438 | (H)Arg-Glu-Phe-Arg-kbt)
Affinity DataKi:  31nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed