Affinity DataKi: 15nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Affinity on 5-hydroxytryptamine 2 receptor labeled by [125I]DOIMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to 5-hydroxytryptamine 2 receptor in rat frontal cortical membranes by [3H]- KET displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor using [125I]DOI as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Compound was evaluated for binding affinity towards 5-hydroxytryptamine 2 receptor in rat anterior cortex using [125I]DOI as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Compound was evaluated for binding affinity towards 5-hydroxytryptamine 2 receptor in rat anterior cortex using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor using [3H]ket as radioligand.More data for this Ligand-Target Pair