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Found 5 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50137628'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50137628(CHEMBL1830682 | CHEMBL60048 | N-(4-(6,7-dimethoxy-...)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor in guinea pig brain after 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Washington University

Curated by ChEMBL
LigandPNGBDBM50137628(CHEMBL1830682 | CHEMBL60048 | N-(4-(6,7-dimethoxy-...)
Affinity DataKi:  3.08E+3nMAssay Description:Displacement of 5-bromo-N-(4-(3,4-dihydro-6,7-dimethoxyisoquinolin-2(1H)-yl)butyl)-2,3-dimethoxybenzamide from sigma-1 receptor in mouse EMT6 cell me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50137628(CHEMBL1830682 | CHEMBL60048 | N-(4-(6,7-dimethoxy-...)
Affinity DataKi:  3.08E+3nMAssay Description:Binding affinity to sigma-1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50137628(CHEMBL1830682 | CHEMBL60048 | N-(4-(6,7-dimethoxy-...)
Affinity DataKi:  3.08E+3nMAssay Description:Binding affinity to sigma-1 opioid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50137628(CHEMBL1830682 | CHEMBL60048 | N-(4-(6,7-dimethoxy-...)
Affinity DataKi:  3.08E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed