Found 3 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50295425'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor in human Jurkat cells after 120 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 223nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 opioid receptor in rat liver homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 223nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat liver membrane by liquid scintillation countingMore data for this Ligand-Target Pair