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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium/glucose cotransporter 2' and Ligand = 'BDBM104500'
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM104500(US8575114, I-12)
Affinity DataIC50:  33nMAssay Description:Inhibition of human SGLT2 expressed in CHOK1 cells assessed as inhibition of [14C]-AMG uptake after 3 hrs by microbeta scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM104500(US8575114, I-12)
Affinity DataIC50:  36.6nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In DepthDetails US Patent