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Found 1 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 2 subunit alpha' and Ligand = 'BDBM154245'
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM154245(US9012443, 261)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of 20% inactivated human Nav1.2 expressed in CHO cells assessed as inhibition of peak inward current by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed