Found 4 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent GABA transporter 1' and Ligand = 'BDBM50063511' TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 3.89E+3nMAssay Description:Binding affinity to mouse GAT1 expressed in HEK293 cells using NO71156 as unlabelled marker by LC-ESI-MS-MS based competitive MS binding assayMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Binding affinity to human GAT1 expressed in HEK293 cells using NO71156 as unlabelled marker by LC-ESI-MS-MS based competitive MS binding assayMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of human GAT1 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
