Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent GABA transporter 2' and Ligand = 'BDBM50427387'
TargetSodium- and chloride-dependent GABA transporter 2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50427387(CHEMBL2326025)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT3 expressed in HEK293 cells after 3 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50427387(CHEMBL2326025)
Affinity DataIC50:  7.59E+5nMAssay Description:Inhibition of mouse mGAT3 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake after 3 mins incubation by TopCount microplate scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50427387(CHEMBL2326025)
Affinity DataIC50:  7.65E+5nMAssay Description:Inhibition of mouse mGAT3 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake after 3 mins incubation by TopCount microplate scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50427387(CHEMBL2326025)
Affinity DataIC50:  7.65E+5nMAssay Description:Inhibition of mouse mGAT3 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake after 3 mins incubation by TopCount microplate scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50427387(CHEMBL2326025)
Affinity DataIC50:  7.65E+5nMAssay Description:Inhibition of mouse mGAT3 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake after 3 mins incubation by TopCount microplate scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed